Publications & Works

Publication Network
Articles 14
All (14)
SCI-E, SSCI, AHCI (11)
SCI-E, SSCI, AHCI, ESCI (13)
ESCI (2)
Scopus (13)
TRDizin (3)

1. Novel benzenesulfonamide-Thiourea derivatives as potent carbonic anhydrase inhibitors with anticancer activity

TRAWALLY M., DEMİR YAZICI K., ARCAN G. G., Vullo D., AKSOY SAĞIRLI P., AKDEMİR A., et al.
JOURNAL OF SULFUR CHEMISTRY , 2026 (SCI-Expanded, Scopus) identifier

2. Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies

Demir Yazıcı K., Trawally M., Bua S., Öztürk-Civelek D., Akdemir A., Supuran C. T., et al.
Bioorganic Chemistry , vol.144, 2024 (SCI-Expanded, Scopus) Sustainable Development identifier identifier identifier

3. Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies

Trawally M., DEMİR YAZICI K., Angeli A., Kaya K., Akdemir A., Supuran C. T., et al.
Anti-Cancer Agents in Medicinal Chemistry , vol.24, no.9, pp.649-667, 2024 (SCI-Expanded, Scopus) Sustainable Development identifier identifier identifier

4. Dithiocarbamates and dithiocarbonates containing 6-nitrosaccharin scaffold: Synthesis, antimycobacterial activity and in silico target prediction using ensemble docking-based reverse virtual screening

Trawally M., Demir Yazıcı K., İpek Dingiş-Birgül S., Kaya K., Akdemir A., Güzel Akdemir Ö.
Journal of Molecular Structure , vol.1277, 2023 (SCI-Expanded, Scopus) Sustainable Development identifier identifier

5. Evaluation of some o-benzenedisulfonimido– sulfonamide derivatives as potent antimicrobial agents

Demir Yazıcı K., Yılmaz F. N., Özbek Çelik B., Güzel Akdemir Ö.
Istanbul Journal of Pharmacy , vol.52, no.3, pp.297-301, 2022 (TRDizin)

6. Mandelic acid-based spirothiazolidinones targeting M. tuberculosis: Synthesis, in vitro and in silico investigations

Trawally M., Demir-Yazici K., Dingiş Birgül S. İ., Kaya K., Akdemir A., Güzel-Akdemir Ö.
BIOORGANIC CHEMISTRY , vol.121, 2022 (SCI-Expanded, Scopus) Sustainable Development identifier identifier identifier

7. Synthesis and potential antitumor activities of mandelic acid linked 2-aryl-1,3-thiazolidin-4-ones

Demir-Yazici K., Guzel-Akdemir O.
JOURNAL OF RESEARCH IN PHARMACY , vol.26, no.4, pp.931-940, 2022 (ESCI) Sustainable Development identifier identifier identifier

8. New Pyridinium Salt Derivatives of 2-(Hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide as Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase Isoforms IX and XII

Güzel Akdemir Ö., Demir Yazıcı K., Vullo D., Supuran C. T., Akdemir A.
Anti-Cancer Agents in Medicinal Chemistry , vol.22, no.14, pp.2637-2646, 2022 (SCI-Expanded, Scopus) identifier identifier identifier

9. Synthesis, molecular modeling and cholinesterase inhibitory effects of 2-indolinone-based hydrazinecarbothioamides

DEMİR YAZICI K., APAYDIN Ç. B., Soylu-Eter O., Ozsoy N., KARALI N. L.
FUTURE MEDICINAL CHEMISTRY , vol.13, no.24, pp.2133-2151, 2021 (SCI-Expanded, Scopus) Sustainable Development identifier identifier identifier

10. Novel Indole-Based Hydrazones as Potent Inhibitors of the alpha-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae

Demir-Yazici K., Guzel-Akdemir Ö., Angeli A., Supuran C. T., Akdemir A.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.21, 2020 (SCI-Expanded) Sustainable Development identifier identifier identifier

11. Development of Thiazolidinones as Fungal Carbonic Anhydrase Inhibitors

Guezel-Akdemir Ö., Carradori S., Grande R., Demir-Yazici K., Angeli A., Supuran C. T., et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.21, no.8, 2020 (SCI-Expanded, Scopus) identifier identifier identifier

12. Evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidin-3-yl)-2-phenylacetamide derivatives as potential antimycobacterial agents

GÜZEL AKDEMİR Ö., DEMİR YAZICI K., TRAWALLY M., DİNGİŞ BİRGÜL S. İ., Akdemir A.
Organic Communications , vol.13, no.2, pp.33-50, 2020 (ESCI, Scopus, TRDizin) identifier identifier

13. Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII

Demir-Yazici K., Bua S., Akgunes N. M., Akdemir A., Supuran C. T., Guzel-Akdemir O.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.20, 2019 (SCI-Expanded, Scopus) identifier identifier identifier

14. Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

Guzel-Akdemir O., Angeli A., Demir K., Supuran C. T., AKDEMİR A.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY , vol.33, no.1, pp.1299-1308, 2018 (SCI-Expanded, Scopus) identifier identifier identifier
Papers Presented at Peer-Reviewed Scientific Conferences 26

1. Unveiling IL11RA variants in craniosynostosis and dental anomalies: insights from exome sequencing

KARAMAN V., Yucesoy M. A., DEMİR YAZICI K., Toksoy G., Yıldız E., KARA B., et al.
58th Conference of the European-Society-of-Human-Genetics (ESHG), Milan, Italy, 24 - 27 May 2025, vol.33, pp.675, (Summary Text) identifier

2. Tail Elongation of OG-001 Enhances Selectivity Toward Tumor-Associated hCA IX and XII

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö.
XII BrazMedChem 2025, Rio De Janeiro, Brazil, 20 - 24 September 2025, pp.1, (Full Text)

3. Structural Simplification of OG-001: Phenyl-to-methyl Substitution Improves Selectivity for Tumor-associated hCA IX and hCA XII

Uzunalioğlu C., Demir Yazıcı K., Trawally M., Akdemir A., Supuran C. T., Güzel Akdemir Ö.
13th Conference on Carbonic Anhydrases (ICCA 2025), Sevilla, Spain, 2 - 04 April 2025, pp.69, (Summary Text)

4. Thione or Thiol: Sructural Confirmation of (E)-2-(1-(4-cyanophenyl)ethylidene)-N-(2-fluoro-4-sulfamoylphenyl)hydrazine-1-Carbothioamide and Carbonic Anhydrase Inhibition Studies

Guliyeva L., Trawally M., Demir-Yazıcı K., Kaya K., Akdemir A., Güzel-Akdemir Ö.
8th International Students Science Congress, İzmir, Turkey, 23 - 24 May 2024, pp.141, (Summary Text)

5. Thione or Thiol: Structural Confirmation of (E)-2-(1-(4-cyanophenyl)ethylidene)-N-(2-fluoro-4-sulfamoylphenyl)hydrazine-1-carbothioamide and Carbonic Anhydrase Inhibition Studies

Guliyeva L., DEMİR YAZICI K., TRAWALLY M., KAYA K., AKDEMİR A., GÜZEL AKDEMİR Ö.
8th International Students Science Congress, İzmir, Turkey, 23 - 24 May 2024, (Summary Text)

6. Synthesis, FTIR spectrum, experimental and theoretical crystal studies, and carbonic anhydrase inhibition studies on 2-[(1H-Pyrrol-2-yl)methylidene]-N-(3-sulfamoylphenyl)hydrazine-1-carbothioamide

TRAWALLY M., DEMİR YAZICI K., KAYA K., AKDEMİR A., GÜZEL AKDEMİR Ö.
12th Internation Drug Chemistry Conferences, Antalya, Turkey, 07 March 2024, (Summary Text)

7. Modification of SLC-0111 as Novel Carbonic Anhydrase Inhibitors

Guliyeva L., M. T., DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Physics, Baku, Azerbaijan, 30 November 2023, (Summary Text)

8. Development of Selective Inhibitors for the Tumor-Associated Carbonic Anhydrases

AKDEMİR A., DEMİR YAZICI K., M. T., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Physics, Baku, Azerbaijan, 30 November 2023, (Summary Text)

9. Modification of SLC-0111 as Novel Carbonic Anhydrse Inhibitors

Guliyeva L., TRAWALLY M., DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Pyhsics, Baku, Azerbaijan, 30 November - 01 December 2023, (Summary Text)

10. Molecular Modeling Studies on Dithiocarbamates and Dithiocarbonates Containing 6-nitrosaccharin Scaffold as antitubercular agents

DİNGİŞ BİRGÜL S. İ., M. T., DEMİR YAZICI K., GÜZEL AKDEMİR Ö., AKDEMİR A.
10th Internation Drug Chemistry Conferences, Turkey, 10 March 2022, (Full Text)

11. Novel sulfa drug containing thiourea derivatives: Synthesis, molecular modelling and inhibition studies of pharmaceutically important carbonic anhydrase isoforms

M. T., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Turkey, 10 - 13 March 2023, (Full Text)

12. Novel sulfa drug containing thiourea derivatives: Synthesis, molecular modelling and inhibition studies pharmaceutical important carbonic anhydrase isoforms

Trawally M., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Antalya, Turkey, 10 - 13 March 2022, pp.27-30, (Full Text)

13. Molecular modelling studies on dithiocarbamates and dithiocarbonates containing 6-nitrosaccharin scaffold as antitubercular agents

DİNGİŞ BİRGÜL S. İ., Trawally M., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Kemer, Antalya, Antalya, Turkey, 10 - 13 March 2022, pp.33-36, (Full Text)

14. SYNTHESIS AND HUMAN CARBONIC ANHYDRASE INHIBITION STUDIES OF SOME 1,3,4-THIADIAZOLES

Demir Yazıcı K., Güzel Akdemir Ö.
13th International Symposium on Pharmaceutical Sciences (ISOPS), Ankara, Turkey, 22 - 25 June 2021, pp.309, (Full Text)

15. Mandelic acid-based novel spirothiazolidinones: Synthesis, antimycobacterial activity and molecular modelling studies

M. T., DEMİR YAZICI K., DİNGİŞ BİRGÜL S. İ., GÜZEL AKDEMİR Ö., AKDEMİR A.
13th International Symposium on Pharmaceutical Sciences, 22 - 24 June 2021, (Full Text)

16. Synthesis and Human Carbonıc Anhydrase Inhıbition Studies of Some 1,3,4-Thiadiazoles

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
İSOPS 13 International Symposium on Pharmaceutical Sciences, Ankara, Turkey, 22 - 25 June 2021, (Full Text)

17. NOVEL THIOSEMICARBAZONES-BASED BENZENESULFONAMIDE hCAII INHIBITORS: SYNTHESIS, BIOLOGICAL EVALUATION AND DOCKING STUDIES

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö., Akdemir A.
3rd INTERNATIONAL AFRICAN CONFERENCE ON CURRENT STUDIES, 27 February - 28 August 2021, pp.718, (Summary Text)

18. Synthesis and Inhibitory Activity of 2-(alkylidene/arylidene)-N-(2-(non) substituted-3/4-sulfamoylphenyl)hydrazine-1-carbothioamide Derivatives Tumor-Associated Carbonic Anhydrase hCA IX and hCA XII Inhibitors

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö.
8th Internation Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.235, (Summary Text)

19. Inhibition of the α-class Carbonic Anhydrase from Vibrio cholera(VchCA) with Novel Sulfonamido based Hydrozones

Güzel Akdemir Ö., Demir Yazıcı K.
8th Interntional Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.69, (Full Text)

20. The Ongoing Quest for Selective hCA IX/XII Inhibitors

Güzel Akdemir Ö., Trawally M., Demir Yazıcı K., Akdemir A., Angeli A., Supuran C. T.
8th Internation Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.307, (Summary Text)

21. Inhibition of the α-class Carbonic Anhydrase from Vibrio cholerae (VchCA) with Novel Sulfonamido-based Hydrazones

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th Internation Drug Chemistry Conferences, 27 February - 01 March 2020, (Full Text)

22. Design, Synthesis and Anticancer Activity of 2-(Hydrazinocarbonyl)-3-Phenyl-1H-Indole-5-Sulfonamide Based Thiosemicarbazides

Demir Yazıcı K., Bua S., Nocentini A., Akdemir A., Supuran C., Güzel Akdemir Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, Italy, 14 - 17 November 2019, pp.27, (Full Text)

23. Design and synthesis of novel indole based hydrazones containing sulfonamide moiety as selective inhibitors of tumour-associated carbonic anhydrase isoforms IX and XII

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, Italy, 14 - 17 November 2019, vol.1, no.1, pp.10, (Full Text)

24. New Sulfonamidoindole Based Hydrazones as Potent and Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase IX and XII Isoforms

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, Italy, 14 - 17 November 2019, vol.1, no.1, pp.11, (Full Text)

25. Tiyazolidinon iskeleti taşıyan bazı yeni bileşiklerin sentezi, yapılarının aydınlatılması ve antikanser aktivitelerinin incelenmesi

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
2. Ulusal Marmara Eczacılık Kongresi (UMEK-2018), İstanbul, Turkey, 14 - 16 November 2018, pp.111, (Summary Text)

26. Molecular modelling studies to guide synthesis programs of new thiourea compounds as putative inhibitors of hCA IX/XII and VcCA.

DEMİR K., Güzel Akdemir Ö., Karalı N. L., Akdemir A.
3rd Satellite Meeting on Carbonic Anhydrase, Montecatini Terme, Italy, 24 - 27 May 2017, pp.68, (Full Text)
Metrics

Publication

40

Publication (WoS)

14

Publication (Scopus)

13

Citation (WoS)

113

H-Index (WoS)

7

Citation (Scopus)

129

H-Index (Scopus)

7

Citation (TrDizin)

1

H-Index (TrDizin)

1

Citation (Sobiad)

8

H-Index (Sobiad)

1

Citation (Sum Other)

1

Project

9

Open Access

5
UN Sustainable Development Goals