Yayınlar & Eserler

Yayın Ağı
Makaleler 13
Tümü (13)
SCI-E, SSCI, AHCI (10)
SCI-E, SSCI, AHCI, ESCI (12)
ESCI (2)
Scopus (12)
TRDizin (3)

1. Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies

Demir Yazıcı K., Trawally M., Bua S., Öztürk-Civelek D., Akdemir A., Supuran C. T., et al.
Bioorganic Chemistry , cilt.144, 2024 (SCI-Expanded, Scopus) Sürdürülebilir Kalkınma identifier identifier identifier

2. Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies

Trawally M., DEMİR YAZICI K., Angeli A., Kaya K., Akdemir A., Supuran C. T., et al.
Anti-Cancer Agents in Medicinal Chemistry , cilt.24, sa.9, ss.649-667, 2024 (SCI-Expanded, Scopus) Sürdürülebilir Kalkınma identifier identifier identifier

3. Dithiocarbamates and dithiocarbonates containing 6-nitrosaccharin scaffold: Synthesis, antimycobacterial activity and in silico target prediction using ensemble docking-based reverse virtual screening

Trawally M., Demir Yazıcı K., İpek Dingiş-Birgül S., Kaya K., Akdemir A., Güzel Akdemir Ö.
Journal of Molecular Structure , cilt.1277, 2023 (SCI-Expanded, Scopus) Sürdürülebilir Kalkınma identifier identifier

4. Evaluation of some o-benzenedisulfonimido– sulfonamide derivatives as potent antimicrobial agents

Demir Yazıcı K., Yılmaz F. N., Özbek Çelik B., Güzel Akdemir Ö.
Istanbul Journal of Pharmacy , cilt.52, sa.3, ss.297-301, 2022 (Hakemli Dergi)

5. Mandelic acid-based spirothiazolidinones targeting M. tuberculosis: Synthesis, in vitro and in silico investigations

Trawally M., Demir-Yazici K., Dingiş Birgül S. İ., Kaya K., Akdemir A., Güzel-Akdemir Ö.
BIOORGANIC CHEMISTRY , cilt.121, 2022 (SCI-Expanded, Scopus) Sürdürülebilir Kalkınma identifier identifier identifier

6. New Pyridinium Salt Derivatives of 2-(Hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide as Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase Isoforms IX and XII

Güzel Akdemir Ö., Demir Yazıcı K., Vullo D., Supuran C. T., Akdemir A.
Anti-Cancer Agents in Medicinal Chemistry , cilt.22, sa.14, ss.2637-2646, 2022 (SCI-Expanded) identifier identifier identifier

7. Synthesis and potential antitumor activities of mandelic acid linked 2-aryl-1,3-thiazolidin-4-ones

Demir-Yazici K., Guzel-Akdemir O.
JOURNAL OF RESEARCH IN PHARMACY , cilt.26, sa.4, ss.931-940, 2022 (ESCI) Sürdürülebilir Kalkınma identifier identifier identifier

8. Synthesis, molecular modeling and cholinesterase inhibitory effects of 2-indolinone-based hydrazinecarbothioamides

DEMİR YAZICI K., APAYDIN Ç. B., Soylu-Eter O., Ozsoy N., KARALI N. L.
FUTURE MEDICINAL CHEMISTRY , cilt.13, sa.24, ss.2133-2151, 2021 (SCI-Expanded) Sürdürülebilir Kalkınma identifier identifier identifier

9. Novel Indole-Based Hydrazones as Potent Inhibitors of the alpha-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae

Demir-Yazici K., Guzel-Akdemir Ö., Angeli A., Supuran C. T., Akdemir A.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , cilt.21, 2020 (SCI-Expanded) Sürdürülebilir Kalkınma identifier identifier identifier

10. Development of Thiazolidinones as Fungal Carbonic Anhydrase Inhibitors

Guezel-Akdemir Ö., Carradori S., Grande R., Demir-Yazici K., Angeli A., Supuran C. T., et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , cilt.21, sa.8, 2020 (SCI-Expanded, Scopus) identifier identifier identifier

11. Evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidin-3-yl)-2-phenylacetamide derivatives as potential antimycobacterial agents

GÜZEL AKDEMİR Ö., DEMİR YAZICI K., TRAWALLY M., DİNGİŞ BİRGÜL S. İ., Akdemir A.
Organic Communications , cilt.13, sa.2, ss.33-50, 2020 (ESCI, Scopus, TRDizin) identifier identifier

12. Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII

Demir-Yazici K., Bua S., Akgunes N. M., Akdemir A., Supuran C. T., Guzel-Akdemir O.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , cilt.20, 2019 (SCI-Expanded, Scopus) identifier identifier identifier

13. Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

Guzel-Akdemir O., Angeli A., Demir K., Supuran C. T., AKDEMİR A.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY , cilt.33, sa.1, ss.1299-1308, 2018 (SCI-Expanded) identifier identifier identifier
Hakemli Bilimsel Toplantılarda Yayımlanmış Bildiriler 25

1. Tail Elongation of OG-001 Enhances Selectivity Toward Tumor-Associated hCA IX and XII

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö.
XII BrazMedChem 2025, Rio De Janeiro, Brezilya, 20 - 24 Eylül 2025, ss.1, (Tam Metin Bildiri)

2. Structural Simplification of OG-001: Phenyl-to-methyl Substitution Improves Selectivity for Tumor-associated hCA IX and hCA XII

Uzunalioğlu C., Demir Yazıcı K., Trawally M., Akdemir A., Supuran C. T., Güzel Akdemir Ö.
13th Conference on Carbonic Anhydrases (ICCA 2025), Sevilla, İspanya, 2 - 04 Nisan 2025, ss.69, (Özet Bildiri)

3. Thione or Thiol: Sructural Confirmation of (E)-2-(1-(4-cyanophenyl)ethylidene)-N-(2-fluoro-4-sulfamoylphenyl)hydrazine-1-Carbothioamide and Carbonic Anhydrase Inhibition Studies

Guliyeva L., Trawally M., Demir-Yazıcı K., Kaya K., Akdemir A., Güzel-Akdemir Ö.
8th International Students Science Congress, İzmir, Türkiye, 23 - 24 Mayıs 2024, ss.141, (Özet Bildiri)

4. Thione or Thiol: Structural Confirmation of (E)-2-(1-(4-cyanophenyl)ethylidene)-N-(2-fluoro-4-sulfamoylphenyl)hydrazine-1-carbothioamide and Carbonic Anhydrase Inhibition Studies

Guliyeva L., DEMİR YAZICI K., TRAWALLY M., KAYA K., AKDEMİR A., GÜZEL AKDEMİR Ö.
8th International Students Science Congress, İzmir, Türkiye, 23 - 24 Mayıs 2024, (Özet Bildiri)

5. Synthesis, FTIR spectrum, experimental and theoretical crystal studies, and carbonic anhydrase inhibition studies on 2-[(1H-Pyrrol-2-yl)methylidene]-N-(3-sulfamoylphenyl)hydrazine-1-carbothioamide

TRAWALLY M., DEMİR YAZICI K., KAYA K., AKDEMİR A., GÜZEL AKDEMİR Ö.
12th Internation Drug Chemistry Conferences, Antalya, Türkiye, 07 Mart 2024, (Özet Bildiri)

6. Modification of SLC-0111 as Novel Carbonic Anhydrase Inhibitors

Guliyeva L., M. T., DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Physics, Baku, Azerbaycan, 30 Kasım 2023, (Özet Bildiri)

7. Development of Selective Inhibitors for the Tumor-Associated Carbonic Anhydrases

AKDEMİR A., DEMİR YAZICI K., M. T., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Physics, Baku, Azerbaycan, 30 Kasım 2023, (Özet Bildiri)

8. Modification of SLC-0111 as Novel Carbonic Anhydrse Inhibitors

Guliyeva L., TRAWALLY M., DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th International Conference Modern Trends in Pyhsics, Baku, Azerbaycan, 30 Kasım - 01 Aralık 2023, (Özet Bildiri)

9. Molecular Modeling Studies on Dithiocarbamates and Dithiocarbonates Containing 6-nitrosaccharin Scaffold as antitubercular agents

DİNGİŞ BİRGÜL S. İ., M. T., DEMİR YAZICI K., GÜZEL AKDEMİR Ö., AKDEMİR A.
10th Internation Drug Chemistry Conferences, Türkiye, 10 Mart 2022, (Tam Metin Bildiri)

10. Novel sulfa drug containing thiourea derivatives: Synthesis, molecular modelling and inhibition studies of pharmaceutically important carbonic anhydrase isoforms

M. T., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Türkiye, 10 - 13 Mart 2023, (Tam Metin Bildiri)

11. Novel sulfa drug containing thiourea derivatives: Synthesis, molecular modelling and inhibition studies pharmaceutical important carbonic anhydrase isoforms

Trawally M., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Antalya, Türkiye, 10 - 13 Mart 2022, ss.27-30, (Tam Metin Bildiri)

12. Molecular modelling studies on dithiocarbamates and dithiocarbonates containing 6-nitrosaccharin scaffold as antitubercular agents

DİNGİŞ BİRGÜL S. İ., Trawally M., DEMİR YAZICI K., AKDEMİR A., GÜZEL AKDEMİR Ö.
10th Internation Drug Chemistry Conferences, Kemer, Antalya, Antalya, Türkiye, 10 - 13 Mart 2022, ss.33-36, (Tam Metin Bildiri)

13. SYNTHESIS AND HUMAN CARBONIC ANHYDRASE INHIBITION STUDIES OF SOME 1,3,4-THIADIAZOLES

Demir Yazıcı K., Güzel Akdemir Ö.
13th International Symposium on Pharmaceutical Sciences (ISOPS), Ankara, Türkiye, 22 - 25 Haziran 2021, ss.309, (Tam Metin Bildiri)

14. Mandelic acid-based novel spirothiazolidinones: Synthesis, antimycobacterial activity and molecular modelling studies

M. T., DEMİR YAZICI K., DİNGİŞ BİRGÜL S. İ., GÜZEL AKDEMİR Ö., AKDEMİR A.
13th International Symposium on Pharmaceutical Sciences, 22 - 24 Haziran 2021, (Tam Metin Bildiri)

15. Synthesis and Human Carbonıc Anhydrase Inhıbition Studies of Some 1,3,4-Thiadiazoles

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
İSOPS 13 International Symposium on Pharmaceutical Sciences, Ankara, Türkiye, 22 - 25 Haziran 2021, (Tam Metin Bildiri)

16. NOVEL THIOSEMICARBAZONES-BASED BENZENESULFONAMIDE hCAII INHIBITORS: SYNTHESIS, BIOLOGICAL EVALUATION AND DOCKING STUDIES

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö., Akdemir A.
3rd INTERNATIONAL AFRICAN CONFERENCE ON CURRENT STUDIES, 27 Şubat - 28 Ağustos 2021, ss.718, (Özet Bildiri)

17. The Ongoing Quest for Selective hCA IX/XII Inhibitors

Güzel Akdemir Ö., Trawally M., Demir Yazıcı K., Akdemir A., Angeli A., Supuran C. T.
8th Internation Drug Chemistry Conference, Antalya, Türkiye, 27 Şubat - 01 Mart 2020, ss.307, (Özet Bildiri)

18. Inhibition of the α-class Carbonic Anhydrase from Vibrio cholera(VchCA) with Novel Sulfonamido based Hydrozones

Güzel Akdemir Ö., Demir Yazıcı K.
8th Interntional Drug Chemistry Conference, Antalya, Türkiye, 27 Şubat - 01 Mart 2020, ss.69, (Tam Metin Bildiri)

19. Synthesis and Inhibitory Activity of 2-(alkylidene/arylidene)-N-(2-(non) substituted-3/4-sulfamoylphenyl)hydrazine-1-carbothioamide Derivatives Tumor-Associated Carbonic Anhydrase hCA IX and hCA XII Inhibitors

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö.
8th Internation Drug Chemistry Conference, Antalya, Türkiye, 27 Şubat - 01 Mart 2020, ss.235, (Özet Bildiri)

20. Inhibition of the α-class Carbonic Anhydrase from Vibrio cholerae (VchCA) with Novel Sulfonamido-based Hydrazones

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
8th Internation Drug Chemistry Conferences, 27 Şubat - 01 Mart 2020, (Tam Metin Bildiri)

21. Design, Synthesis and Anticancer Activity of 2-(Hydrazinocarbonyl)-3-Phenyl-1H-Indole-5-Sulfonamide Based Thiosemicarbazides

Demir Yazıcı K., Bua S., Nocentini A., Akdemir A., Supuran C., Güzel Akdemir Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, İtalya, 14 - 17 Kasım 2019, ss.27, (Tam Metin Bildiri)

22. Design and synthesis of novel indole based hydrazones containing sulfonamide moiety as selective inhibitors of tumour-associated carbonic anhydrase isoforms IX and XII

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, İtalya, 14 - 17 Kasım 2019, cilt.1, sa.1, ss.10, (Tam Metin Bildiri)

23. New Sulfonamidoindole Based Hydrazones as Potent and Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase IX and XII Isoforms

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.
4th Satellite International Meeting on Carbonic Anhydrase, Parma, İtalya, 14 - 17 Kasım 2019, cilt.1, sa.1, ss.11, (Tam Metin Bildiri)

24. Tiyazolidinon iskeleti taşıyan bazı yeni bileşiklerin sentezi, yapılarının aydınlatılması ve antikanser aktivitelerinin incelenmesi

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.
2. Ulusal Marmara Eczacılık Kongresi (UMEK-2018), İstanbul, Türkiye, 14 - 16 Kasım 2018, ss.111, (Özet Bildiri)

25. Molecular modelling studies to guide synthesis programs of new thiourea compounds as putative inhibitors of hCA IX/XII and VcCA.

DEMİR K., Güzel Akdemir Ö., Karalı N. L., Akdemir A.
3rd Satellite Meeting on Carbonic Anhydrase, Montecatini Terme, İtalya, 24 - 27 Mayıs 2017, ss.68, (Tam Metin Bildiri)
Metrikler

Yayın

38

Yayın (WoS)

12

Yayın (Scopus)

12

Atıf (WoS)

114

H-İndeks (WoS)

5

Atıf (Scopus)

129

H-İndeks (Scopus)

7

Atıf (TrDizin)

1

H-İndeks (TrDizin)

1

Atıf (Sobiad)

8

H-İndeks (Sobiad)

1

Atıf (Diğer Toplam)

1

Proje

9

Açık Erişim

5
BM Sürdürülebilir Kalkınma Amaçları