Prof. Özlen GÜZEL AKDEMİR

Publication Network

Published journal articles indexed by SCI, SSCI, and AHCI

Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies

Demir Yazıcı K., Trawally M., Bua S., Öztürk-Civelek D., Akdemir A., Supuran C. T., et al.

Bioorganic Chemistry , vol.144, 2024 (SCI-Expanded) Sustainable Development

Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies

Trawally M., DEMİR YAZICI K., Angeli A., Kaya K., Akdemir A., Supuran C. T., et al.

Anti-Cancer Agents in Medicinal Chemistry , vol.24, no.9, pp.649-667, 2024 (SCI-Expanded)

Urease inhibitors for the treatment of H. pylori

GÜZEL AKDEMİR Ö., Akdemir A.

Expert Opinion on Therapeutic Patents , 2024 (SCI-Expanded)

Dithiocarbamates and dithiocarbonates containing 6-nitrosaccharin scaffold: Synthesis, antimycobacterial activity and in silico target prediction using ensemble docking-based reverse virtual screening

Trawally M., Demir Yazıcı K., İpek Dingiş-Birgül S., Kaya K., Akdemir A., Güzel Akdemir Ö.

Journal of Molecular Structure , vol.1277, 2023 (SCI-Expanded) Sustainable Development

Mandelic acid-based spirothiazolidinones targeting M. tuberculosis: Synthesis, in vitro and in silico investigations

Trawally M., Demir-Yazici K., Dingiş Birgül S. İ., Kaya K., Akdemir A., Güzel-Akdemir Ö.

BIOORGANIC CHEMISTRY , vol.121, 2022 (SCI-Expanded) Sustainable Development

New Pyridinium Salt Derivatives of 2-(Hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide as Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase Isoforms IX and XII

Güzel Akdemir Ö., Demir Yazıcı K., Vullo D., Supuran C. T., Akdemir A.

Anti-Cancer Agents in Medicinal Chemistry , vol.22, no.14, pp.2637-2646, 2022 (SCI-Expanded)

Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII

Akocak S., Guzel-Akdemir O., Sanku R. K. K., Russom S. S., Iorga B. I., Supuran C. T., et al.

BIOORGANIC CHEMISTRY , vol.103, 2020 (SCI-Expanded)

Synthesis and antibacterial activity of new hybrid derivatives of 5-sulfamoyl-1H-indole and 4-thiazolidinone groups

Guzel-Akdemir O., Trawally M., Ozbek-Babuc M., Ozbek-Celik B., Ermut G., Ozdemir H.

MONATSHEFTE FUR CHEMIE , vol.151, pp.1443-1452, 2020 (SCI-Expanded)

Novel Indole-Based Hydrazones as Potent Inhibitors of the alpha-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae

Demir-Yazici K., Guzel-Akdemir Ö., Angeli A., Supuran C. T., Akdemir A.

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.21, 2020 (SCI-Expanded) Sustainable Development

Development of Thiazolidinones as Fungal Carbonic Anhydrase Inhibitors

Guezel-Akdemir Ö., Carradori S., Grande R., Demir-Yazici K., Angeli A., Supuran C. T., et al.

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.21, no.8, 2020 (SCI-Expanded)

Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII

Demir-Yazici K., Bua S., Akgunes N. M., Akdemir A., Supuran C. T., Guzel-Akdemir O.

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES , vol.20, 2019 (SCI-Expanded)

Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

Guzel-Akdemir O., Angeli A., Demir K., Supuran C. T., AKDEMİR A.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY , vol.33, no.1, pp.1299-1308, 2018 (SCI-Expanded)

Isatin analogs as novel inhibitors of Candida spp. beta-carbonic anhydrase enzymes

Akdemir A., Guzel-Akdemir O., Karali N. L., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.24, no.8, pp.1648-1652, 2016 (SCI-Expanded)

Discovery of novel isatin-based sulfonamides with potent and selective inhibition of the tumor-associated carbonic anhydrase isoforms IX and XII

Guzel-Akdemir O., AKDEMİR A., Karali N., Supuran C. T.

ORGANIC & BIOMOLECULAR CHEMISTRY , vol.13, no.23, pp.6493-6499, 2015 (SCI-Expanded)

Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition

Guzel-Akdemir O., Biswas S., Lastra K., McKenna R., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.21, no.21, pp.6674-6680, 2013 (SCI-Expanded)

Inhibition of tumor-associated human carbonic anhydrase isozymes IX and XII by a new class of substituted-phenylacetamido aromatic sulfonamides

AKDEMİR A., Guzel-Akdemir O., Scozzafava A., Capasso C., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.21, no.17, pp.5228-5232, 2013 (SCI-Expanded)

A Class of Sulfonamides with Strong Inhibitory Action against the alpha-Carbonic Anhydrase from Trypanosoma cruzi

Guzel-Akdemir O., AKDEMİR A., Pan P., Vermelho A. B., Parkkila S., Scozzafava A., et al.

JOURNAL OF MEDICINAL CHEMISTRY , vol.56, no.14, pp.5773-5781, 2013 (SCI-Expanded) Sustainable Development

o-Benzenedisulfonimido-sulfonamides are potent inhibitors of the tumor-associated carbonic anhydrase isoforms CA IX and CA XII

Guzel-Akdemir O., Akdemir A., Işık S., Vullo D., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.21, pp.1386-1391, 2013 (SCI-Expanded)

Conformational variability of different sulfonamide inhibitors with thienyl-acetamido moieties attributes to differential binding in the active site of cytosolic human carbonic anhydrase isoforms

Biswas S., Aggarwal M., GÜZEL Ö., Scozzafava A., McKenna R., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.19, 2011 (SCI-Expanded)

Carbonic anhydrase inhibitors. The ß-carbonic anhydrases from the fungal pathogens Cryptococcus neoformans and Candida albicans are strongly inhibited by substituted-phenyl-1H-indole-5-sulfonamides

GÜZEL Ö., Maresca A., Hall R. A., Scozzafava A., Mastrolorenzo A., Mühlschlegel F. A., et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS , vol.20, pp.2508-2511, 2010 (SCI-Expanded)

3-Phenyl-1H-Indole-5-Sulfonamides: Structure-Based Drug Design of a Promising Class of Carbonic Anhydrase Inhibitors

Guzel O., Innocenti A., Vullo D., Scozzafava A., Supuran C. T.

CURRENT PHARMACEUTICAL DESIGN , vol.16, no.29, pp.3317-3326, 2010 (SCI-Expanded) Sustainable Development

Synthesis and biological evaluation of new 4-thiazolidinone derivatives

Guzel O., Salman A.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY , vol.24, no.4, pp.1015-1023, 2009 (SCI-Expanded)

Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitochondrial isoforms VA and VB

Guzel O., Innocenti A., Scozzafava A., Salman A., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.17, no.14, pp.4894-4899, 2009 (SCI-Expanded)

Discovery of Low Nanomolar and Subnanomolar Inhibitors of the Mycobacterial beta-Carbonic Anhydrases Rv1284 and Rv3273

Guzel O., Maresca A., Scozzafava A., Salman A., Balaban A. T., Supuran C. T.

JOURNAL OF MEDICINAL CHEMISTRY , vol.52, no.13, pp.4063-4067, 2009 (SCI-Expanded) Sustainable Development

Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitchondrial isoforms VA and VB

GÜZEL Ö., Innocenti A., Scozzafava A., Salman A., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.17, pp.4894-4899, 2009 (SCI-Expanded)

Carbonic anhydrase inhibitors. Phenacetyl-, pyridylacetyl- and thienylacetyl-substituted aromatic sulfonamides act as potent and selective isoform VII inhibitors

GÜZEL Ö., Innocenti A., Scozzafava A., Salman A., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS , vol.19, pp.3170-3173, 2009 (SCI-Expanded)

Carbonic anhydrase inhibitors. The nematode alpha-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides

Guzel O., Innocenti A., Hall R. A., Scozzafava A., Muhlschlegel F. A., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.17, no.8, pp.3212-3215, 2009 (SCI-Expanded)

Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII

GÜZEL Ö., Maresca A., Scozzafava A., Salman A., Balaban A. T., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS , vol.19, pp.2931-2934, 2009 (SCI-Expanded)

Crystal Structure of 1,1,3-trioxo-2,3-dihydro-1,2-benzisothiazol-2-ylmethyl 4-phenyl Piperazine-1-carbodithioate, C19H19N3O3S3.

AKKURT M., Yalcin S. P., Guzel O., Salman A., BÜYÜKGÜNGÖR O.

ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES , vol.65, 2009 (SCI-Expanded)

Carbonic anhydrase inhibitors. Interaction of 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide with 12 mammalian isoforms: kinetic and X-ray crystallographic studies

GÜZEL Ö., Temperini C., Innocenti A., Scozzafava A., Salman A., Supuran C. T.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS , vol.18, pp.152-158, 2008 (SCI-Expanded)

Synthesis and antituberculosis activity of 5-methyl/trifluoromethoxy-1H-indole-2,3-dione 3-thiosemicarbazone derivatives

Guzel O., Karali N., Salman A.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.16, no.19, pp.8976-8987, 2008 (SCI-Expanded) Sustainable Development

N-(2,6-dimethyl-3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-2-hydroxy-2,2-diphenylacetamide

Yalcin S. P., AKKURT M., ŞAHİN E., Guzel O., Salman A., Ihan E.

ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE , vol.64, 2008 (SCI-Expanded)

Carbonic anhydrase inhibitors. Synthesis and inhibition studies against mammalian isoforms I – XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides

GÜZEL Ö., Innocenti A., Scozzafava A., Salman A., Parkkila S., Hilvo M., et al.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.16, pp.9113-9120, 2008 (SCI-Expanded)

Synthesis and antituberculosis activity of 5-methyl/trifluoromethoxy-1H-indole-2,3-dione-3-thiosemicarbazone derivatives

GÜZEL Ö., Karalı N., Salman A.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.16, pp.8976-8987, 2008 (SCI-Expanded)

Crystal structure of (1,1-dioxido-3-oxo-1,2-benzisothiazol-2(3H)-yl)methyl O-propyl dithiocarbonate

Akkurt M., Yalçın Ş. P., Büyükgüngör O., GÜZEL Ö., Salman A.

ANALYTICAL SCIENCES , vol.24, 2008 (SCI-Expanded)

1,1,3-Trioxo-2,3-dihydro-1,2-benzisothiazol-2-ylmethyl 4-phenylpiperazine-1-carbodithioate

Akkurt M., Yalçın Ş. P., GÜZEL Ö., Salman A., Büyükgüngör O.

Acta Crystallographica , vol.E63, 2007 (SCI-Expanded)

N-(2,6-dimethyl-3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-2-hydroxy-2,2-diphenylacetamide

Yalçın Ş. P., Akkurt M., Şahin E., GÜZEL Ö., Salman A., İlhan E.

Acta Crystallographica , vol.E64, 2007 (SCI-Expanded)

O-Butyl S-(1,1,3-trioksobenz[d]isothiazol-2-yl)methyl dithiocarbonate

Akkurt M., Karaca S., Şahin E., GÜZEL Ö., Salman A.

Acta Crystallographica , vol.E63, 2007 (SCI-Expanded)

2-Hydroxy-N-(3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-2,2-diphenylacetamide.

Akkurt M., Karaca S., Şahin E., GÜZEL Ö., Salman A., İlhan E.

Acta Crystallographica , vol.E63, 2007 (SCI-Expanded)

Synthesis, antimycobacterial and antitumor activities of new (1,1-dioxido-3-oxo-1,2-benzisothiazol-2(3H)-yl)methyl N,N-disubstituted dithiocarbamate/O-alkyldithiocarbonate derivatives

Guzel O., Salman A.

BIOORGANIC & MEDICINAL CHEMISTRY , vol.14, no.23, pp.7804-7815, 2006 (SCI-Expanded) Sustainable Development

Articles Published in Other Journals

Role of human carbonic anhydrase isoforms VA and VB in obesity: Implications, mechanisms, and therapeutic prospects

Kaçmaz M., Trawally M., GÜZEL AKDEMİR Ö.

Journal of Research in Pharmacy , vol.28, no.3, pp.733-748, 2024 (ESCI)

Antiviral Properties of 5-Sulfamoyl-1H-Indole-Linked Spirothiazolidinone Derivatives: A Study on Human Parainfluenza Virus-2

Trawally M., YILMAZ F. N., ÖZBEK ÇELİK B., Akdemir A., GÜZEL AKDEMİR Ö.

Journal of Research in Pharmacy , vol.28, no.1, pp.213-224, 2024 (ESCI)

Evaluation of some o-benzenedisulfonimido– sulfonamide derivatives as potent antimicrobial agents

Demir Yazıcı K., Yılmaz F. N., Özbek Çelik B., Güzel Akdemir Ö.

Istanbul Journal of Pharmacy , vol.52, no.3, pp.297-301, 2022 (Peer-Reviewed Journal)

Synthesis and potential antitumor activities of mandelic acid linked 2-aryl-1,3-thiazolidin-4-ones

Demir-Yazici K., Guzel-Akdemir O.

JOURNAL OF RESEARCH IN PHARMACY , vol.26, no.4, pp.931-940, 2022 (ESCI) Sustainable Development

Benzilic acid based new 2-aryl-1,3-thiazolidin-4-one derivatives: Synthesis and anticancer activity

Güzel Akdemir Ö., Demir-Yazıcı K.

JOURNAL OF RESEARCH IN PHARMACY , vol.25, no.3, pp.305-317, 2021 (ESCI)

Evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidin-3-yl)-2-phenylacetamide derivatives as potential antimycobacterial agents

GÜZEL AKDEMİR Ö., DEMİR YAZICI K., TRAWALLY M., DİNGİŞ BİRGÜL S. İ., Akdemir A.

Organic Communications , vol.13, no.2, pp.33-50, 2020 (ESCI)

Antimicrobial and antiviral activity of spiroindolinones bearing benzothiazolines moiety

Güzel Ö., Karalı N. L., Ermut G., Birteksöz Tan A. S.

ISTANBUL JOURNAL OF PHARMACY , vol.43, no.1, pp.1-11, 2013 (ESCI)

Spectrophotometric determination of drugs having primary amine group with p-dimethylaminocinnamaldehyde

GÜZEL Ö., Salman A.

TURKİSH JOURNAL OF PHARMACEUTİCAL SCİENCES , vol.4(1), pp.31-39, 2007 (Scopus)

Refereed Congress / Symposium Publications in Proceedings

SYNTHESIS AND HUMAN CARBONIC ANHYDRASE INHIBITION STUDIES OF SOME 1,3,4-THIADIAZOLES

Demir Yazıcı K., Güzel Akdemir Ö.

13th International Symposium on Pharmaceutical Sciences (ISOPS), Ankara, Turkey, 22 - 25 June 2021, pp.309

NOVEL THIOSEMICARBAZONES-BASED BENZENESULFONAMIDE hCAII INHIBITORS: SYNTHESIS, BIOLOGICAL EVALUATION AND DOCKING STUDIES

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö., Akdemir A.

3rd INTERNATIONAL AFRICAN CONFERENCE ON CURRENT STUDIES, 27 February - 28 August 2021, pp.718

Inhibition of the α-class Carbonic Anhydrase from Vibrio cholera(VchCA) with Novel Sulfonamido based Hydrozones

Güzel Akdemir Ö., Demir Yazıcı K.

8th Interntional Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.69

The Ongoing Quest for Selective hCA IX/XII Inhibitors

Güzel Akdemir Ö., Trawally M., Demir Yazıcı K., Akdemir A., Angeli A., Supuran C. T.

8th Internation Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.307

Synthesis and Inhibitory Activity of 2-(alkylidene/arylidene)-N-(2-(non) substituted-3/4-sulfamoylphenyl)hydrazine-1-carbothioamide Derivatives Tumor-Associated Carbonic Anhydrase hCA IX and hCA XII Inhibitors

Trawally M., Demir Yazıcı K., Güzel Akdemir Ö.

8th Internation Drug Chemistry Conference, Antalya, Turkey, 27 February - 01 March 2020, pp.235

New Sulfonamidoindole Based Hydrazones as Potent and Selective Inhibitors of Tumour-Related Human Carbonic Anhydrase IX and XII Isoforms

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.

4th Satellite International Meeting on Carbonic Anhydrase, Parma, Italy, 14 - 17 November 2019, vol.1, no.1, pp.11

Design and synthesis of novel indole based hydrazones containing sulfonamide moiety as selective inhibitors of tumour-associated carbonic anhydrase isoforms IX and XII

DEMİR YAZICI K., Bua S., Akdemir A., Supuran C., GÜZEL AKDEMİR Ö.

4th Satellite International Meeting on Carbonic Anhydrase, Parma, Italy, 14 - 17 November 2019, vol.1, no.1, pp.10

Tiyazolidinon iskeleti taşıyan bazı yeni bileşiklerin sentezi, yapılarının aydınlatılması ve antikanser aktivitelerinin incelenmesi

DEMİR YAZICI K., GÜZEL AKDEMİR Ö.

2. Ulusal Marmara Eczacılık Kongresi (UMEK-2018), İstanbul, Turkey, 14 - 16 November 2018, pp.111

Molecular modelling studies to guide synthesis programs of new thiourea compounds as putative inhibitors of hCA IX/XII and VcCA

Demir K., GÜZEL AKDEMİR Ö., KARALI N. L., AKDEMİR A.

3rd Satellite Meeting on Carbonic Anhydrase, 24 - 27 May 2017, pp.62

Structurally novel thiazolidinone-containing compounds that do not contain sulfonamide groups display antifungal activity

GÜZEL AKDEMİR Ö., Carradori S., Rivanera D., Çapan G., Akdemir A.

3rd Satellite Meeting on Carbonic Anhydrase, Montecatini Terme, Italy, 24 - 27 May 2017, pp.69

Molecular modelling studies to guide synthesis programs of new thiourea compounds as putative inhibitors of hCA IX/XII and VcCA.

DEMİR K., Güzel Akdemir Ö., Karalı N., Akdemir A.

3rd Satellite Meeting on Carbonic Anhydrase, Montecatini Terme, Italy, 24 - 27 May 2017, pp.68

1H-indole-2,3-dione 3-[N-(4-sulfamoylphenyl)thiosemicarbazone] derivatives as putative anticancer and antifungal agents

Akdemir A., KARALI N. L., Supuran C. T., GÜZEL AKDEMİR Ö.

7th European Congress of Pharmacology EPHAR 2016, İstanbul, Turkey, 27 - 30 June 2016, pp.1

Substituted-phenylacetamido aromatic sulfonamides are potent inhibitors of human and Trypanosoma cruzi carbonic anhydrases

GÜZEL AKDEMİR Ö., Akdemir A., Pan P., Vermelho A. B., Parkkila S., Scozzafava A., et al.

10th International Carbonic Anhydrase Conference, Maastricht, Netherlands, 20 - 22 April 2015, pp.48 Sustainable Development

Potent Inhibitors of Mitochondrial Carbonic Anhydrase Isozyme CA-VA and CA-VB and brain associated isozyme CA-VII

Akdemir A., GÜZEL Ö., Supuran C.

9th International Conference on the Carbonic Anhydrases, Antalya, Turkey, 11 - 15 April 2012, pp.67

Pyridinium Derivatives of 3-Aminobenzensulfonamide-Structure-Activity Relationship as Carbonic Anhydrase Inhibitors

Akocak S., GÜZEL Ö., Supuran C., Ilies M. A.

9th International Conference on the Carbonic Anhydrases, Antalya, Turkey, 11 - 15 April 2012, pp.84

5-triflorometoksi-1H-İndol-2,3-Dion 3-Tiyosemikarbazon Türevlerinin Miyeloid, Lenfoid Lösemi Hücreleri ve Akut Lenfoblastik Lösemi Hastalarının Periferik Kan Mononuklear Hücreleri Üzerine Sitotoksik Etkileri.

Çetin M. B., Karadenizli S., Kuruca D. S., Karalı N. L., Güzel Akdemir Ö., Akgün Dar K., et al.

III. Multidisipliner Kanser Araştırma Sempozyumu Teorik Metot Çalıştayı, Bursa, Turkey, 14 - 17 March 2010, pp.40

Carbonic anhydrase inhibitors. The nematode ?-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides

GÜZEL Ö., Innocenti A., Hall R. A., Scozzafava A., Mühlschlegel F. A., Supuran C.

8th International Conference on the Carbonic Anhydrases, Floransa, Italy, 16 - 19 September 2009, pp.43

Synthesis and biological evaluation of new 6-nitrosaccharin derivatives

GÜZEL Ö., Salman A.

9th International Symposium on Pharmaceutical Sciences (ISOPS), Ankara, Turkey, 23 - 26 June 2009, pp.190

Discovery of low nanomolar and subnanomolar inhibitors of the mycobacterial ?-carbonic anhydrases Rv1284 and Rv3273

GÜZEL Ö., Maresca A., Scozzafava A., Salman A., Balaban A. T., Supuran C.

9th International Symposium on Pharmaceutical Sciences (ISOPS), Ankara, Turkey, 23 - 26 June 2009, pp.188

Synthesis and antimycobacterial activity of new 4-thiazolidinone derivatives

GÜZEL AKDEMİR Ö., Salman A., ÇAPAN G.

3rd International Meeting on Medicinal and Pharmaceutical Chemistry, Antalya, Turkey, 16 - 21 October 2007, pp.1

Synthesis of new 4-thiazolidinone derivatives as potential antimycobacterial and antitumor agents

GÜZEL Ö., Salman A.

3rd International Meeting on Medicinal and Pharmaceutical Chemistry (IMMPC-3), Antalya, Turkey, 16 - 21 October 2007, pp.70

Synthesis antimycobacterial and antitumor activities of new5-bromo-N-(3-oxo-1-thia-4-azaspiro[4.4]non-4-yl)/N-(3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-3-phenyl-1H-indole-2-carboxamide derivatives

GÜZEL AKDEMİR Ö., ÇAPAN G., Salman A.

5 th International Symposium on Pharmaceutical Chemistry, İstanbul, Turkey, 5 - 07 September 2007, pp.57

Synthesis, characterization and antituberculosis activity of spiroindolinones

Karalı N., GÜZEL Ö., Salman A.

5th International symposium on Pharmaceutical Chemistry, İstanbul, Turkey, 5 - 07 September 2007, pp.80

Characterization and Antituberculosis Activity of Spiroindolinones

KARALI N. L., GÜZEL Ö., Salman A.

5th International Symposium on Pharmaceutical Chemistry, İstanbul, Turkey, 5 - 07 September 2007, pp.1

One-pot synthesis synthesis of novel substituted 4-(3,4-dimethoxyphenyl)ethyl-1-thia-4-azaspiro[4.5]decan-3-ones

GÜZEL Ö., Terzioğlu N., Gürsoy A.

3rd International Conference on Multi-Component Reactions and Related Chemistry, Amsterdam, Netherlands, 9 - 13 July 2006, pp.87

One-pot synthesis of novel substituted 4-morpholinoethyl-1-thia-4-azaspiro[4.5]decan-3-one

Terzioğlu N., GÜZEL Ö., Gürsoy A.

3rd International Conference on Multi-Component Reactions and Related Chemistry, Amsterdam, Netherlands, 9 - 13 July 2006, pp.129

New 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidin-3-yl)-2-phenylacetamide derivatives: synthesis and antimicrobial evaluation

GÜZEL Ö., Salman A., Terzioğlu N., Çapan G.

2ND International Meeting on Medicinal and Pharmaceutical Chemistry IMMPC-2, Antalya, Turkey, 10 October 2004 - 14 October 2002, pp.141

New 2-hydroxy-N-(4-oxo-2-substitutedphenyl-1,3-thiazolidine-3-yl-2-phenylacetamide derivatives:Synthesis and antimicrobial evaluation

GÜZEL AKDEMİR Ö., Terzioğlu N., Salman A., ÇAPAN G.

2nd International Meeting on Medicinal and Pharmaceutical Chemistry, Antalya, Turkey, 10 - 14 October 2004, pp.141

Synthesis and antimicrobial evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidine-3-yl)-2-phenylacetamide derivatives

GÜZEL AKDEMİR Ö., Salman A., ÇAPAN G.

4th International Symposium on Pharmaceutical Chemistry, İstanbul, Turkey, 17 - 19 September 2003, pp.169

Synthesis and antimicrobial evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3-thiazolidin-3-yl)-2-phenylacetamide derivatives

GÜZEL Ö., Salman A., Çapan G.

4th International Symposium on Pharmaceutical Chemistry, İstanbul, Turkey, 17 September 2003 - 19 September 2002, pp.169-170

Spectrophotometric determination of some drugs incorporating primary amino functions

GÜZEL Ö., Salman A.

1st International Meeting on Medicinal and Pharmaceutical Chemistry IMMPC-1, Ankara, Turkey, 25 - 28 September 2002, pp.78

Synthesis and antimycobacterial activity of new 2-hydroxy-N-(3-oxo-1-thia-4-azaspiro[4.4]non-4-yl)/(3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-2-phenyl-acetamide derivatives

GÜZEL Ö., Çapan G., İlhan E., Salman A.

1st International Meeting on Medicinal and Pharmaceutical Chemistry IMMPC-1, Ankara, Turkey, 25 - 28 September 2002, pp.79

Synthesis and antimicrobial evaluation of new 2-hydroxy-N-(3-oxo-1-thia-4-azaspiro[4.4]non-4yl)/(3-oxo-1-thia-4-azaspiro[4.5]dec-4-yl)-2-phenylacetamide derivatives

GÜZEL AKDEMİR Ö., ÇAPAN G., İlhan E., Salman A.

1st International Meeting on Medicinal and Pharmaceutical Chemistry, Ankara, Turkey, 25 - 28 September 2002, pp.79

Books & Book Chapters

Aromatase

GÜZEL AKDEMİR Ö.

in: Metalloenzymes, Claudiu T. Supuran, William A. Donald, Editor, Academic Press is an imprint of Elsevier, pp.459-464, 2023

Piperine Derivatives: New Trends in Medicinal Chemistry

Trifan A., GÜZEL AKDEMİR Ö., CARRADORİ S.

in: Medicinal Chemistry Lessons From Nature (Volume 3) Alkaloids and Other Nitrogen-Containing Derivatives, Simone Carradori, Editor, Bentham Science Publishers Pte. Ltd. 80 Robinson Road #02-00, Singapore 068898, Singapore2023, pp.100-127, 2023

İlaç Tasarımı: hedef protein ile etkileşim optimizasyonu

GÜZEL AKDEMİR Ö., AKDEMİR A.

in: Medisinal Kimya Giriş, Prof.Dr. Özekin Algül, Editor, Ankara Nobel Tıp Kitapevi, Ankara, pp.223-255, 2021

Antibakteriyel Sülfa İlaçları

GÜZEL AKDEMİR Ö.

in: Medisinal Kimya, Mehmet Alp, Editor, Akademisyen Kitabevi, Ankara, pp.244-264, 2021

Foye Medisinal Kimya Temel İlkeler

GÜZEL AKDEMİR Ö., AKDEMİR A.

Ankara Nobel, 2019

Antipsikotik ve Anksiyolitik İlaçlar

Güzel Akdemir Ö., Akdemir A.

in: Foye Medisinal Kimya Temel İlkeleri, Öztekin Algül,Kayhan Bolelli, Editor, Nobel Yayın Dağıtım, Ankara, pp.96-113, 2019

The Structure, Physiological Role, and Potential Medicinal Applications of Carbonic Anhydrase V

AKDEMİR A., GÜZEL AKDEMİR Ö.

in: Carbonic Anhydrases as Biocatalysts from Theory to Medical and Industrial Applications, Supuran Claudiu, Simone Giuseppina, Editor, Radarweg 29, PO Box 211, 1000 AE Amsterdam, The NetherlandsThe Boulevard, Langford Lane, Kidlington, Oxford OX5 1GB, UK225 Wyman Street, Waltham, MA 02451, USA, pp.125-139, 2015

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